プログラム(ポスター発表の部)

第2日　9月28日(水)

11:10-12:10

ショートプレゼンテーション
Short Presentation
座長：荒井雅吉 (阪大院薬)
Chair: Arai, M. (Graduate School of Pharmaceutical Sciences, Osaka University)

12:10-14:50

ポスター示説
Poster Presentation

P-2

• DPP4阻害活性を有するABT-341のワンポット合成
  • (東理大工)
    ○石川勇人、本間正一、林　雄二郎
• One-Pot Synthesis of the DPP4 Inhibitor ABT-341
  • Ishikawa, H., Honma, M., Hayashi, Y.
    (Department of Engineering, Tokyo University of Science)

P-4

• ¹¹C-標識カプサイシンの合成とPETによるラット体内の分子イメージング
  • (理研分子イメージング)
    ○後藤美樹、水間　広、和田康弘、鈴木正昭、尾上浩隆、渡辺恭良、土居久志
• Synthesis of [¹¹C]Capsaicin and In Vivo PET Study of Rat
  • Goto, M., Mizuma, H., Wada, Y., Suzuki, M., Onoe, H., Watanabe, Y., Doi, H.
    (Center for Molecular Imaging Science, Riken)

P-6

• 金触媒を用いた分子内ヒドロアミノ化反応を基盤としたQuinocarcinの合成研究
  • (京大院薬)
    ○千葉浩亮、大石真也、藤井信孝、大野浩章
• Synthetic Study of Quinocarcin by Au(I)-Catalyzed Intramolecular Hydroamination
  • Chiba, H., Oishi, S., Fujii, N., Ohno, H.
    (Graduate School of Pharmaceutical Sciences, Kyoto University)

P-8

• アトロプルプランの合成研究
  • (東京理大薬)
    ○鈴木孝洋、佐々木　綾、小林　進
• Synthetic Study of Atropurpuran
  • Suzuki, T., Sasaki, A., Kobayashi, S.
    (Faculty of Pharmaceutical Sciences, Tokyo University of Science)

P-10

• 培養細胞によるBiotransformation
  • (弘前大院理工^a、弘前大理工^b、東北大多元研^c)
    長岐正彦^a、○佐藤拓哉^b、木立卓巳^b、田部真吾^c、菊地　陽^a
• Biotransformation by Cultured Cells
  • Nagaki, M.^a, Sato, T.^b, Kidachi, T.^b, Tanabe, S.^c, Kikuchi, Y.^a
    (^aGraduate School of Science and Technology, Hirosaki University, ^bDepartment of Frontier Materials Chemistry, Hirosaki University, ^cIMRAM, Tohoku University)

P-12

• ナトリウムチャネルサブタイプ選択的阻害を志向したサキシトキシン誘導体類の合成と活性評価
  • (東農工大院工^a、東北大院農^b、広島国際大保健医療^c)
    ○秋元隆史^a、篠原涼子^a、岩本　理^a、山下まり^b、山岡　薫^c、長澤和夫^a
• Synthesis of Saxitoxin Derivatives Focusing on the Development of Sodium Channel Subtype Selective Ligands and Evaluation of Their Inhibitory Activity on Sodium Channels
  • Akimoto, T.^a, Shinohara, R.^a, Iwamoto, O.^a, Yotsu-Yamashita, M.^b, Yamaoka, K.^c, Nagasawa, K.^a
    (^aDepartment of Technology, Tokyo University of Agriculture and Technology, ^bDepartment of Agricultural Science, Tohoku University, ^cFaculty of Health Sciences, Hiroshima International University)

P-14

• アジリジンを利用したピロリジン型アルカロイドのエナンチオ選択的合成研究
  • (千葉大院薬)
    ○近藤友香里、熊本卓哉、鈴木紀行、石川　勉
• Enantioselective Synthesis of Pyrrolidine Alkaloids from Aziridine System
  • Kondo, Y., Kumamoto, T., Suzuki, N., Ishikawa, T.
    (Graduate School of Pharmaceutical Sciences, Chiba University)

P-16

• セルラーゼ反応機構解明を目指した反応遷移状態アナログオリゴ糖の合成と評価
  • (弘前大農生^a、長岡技科大^b)
    ○野口翔悟^a、山本和範^a、田邉直哉^a、竹本晋太郎^b、城所俊一^b、橋本　勝^a
• Syntheses of Cellotriose and Cellotetraose Analogues as Transition State Mimics for Mechanistic Studies of Cellulases
  • Noguchi, S.^a, Yamamoto, K.^a, Tanabe, N.^a, Takemoto, S.^b, Kidokoro, S.^b, Hashimoto, M.^a
    (^aAgriculture and Life Science, Hirosaki University, ^bBioengineering, Nagaoka University of Technology)

P-18

• 抗腫瘍性マクロライド化合物amphidinolide B, G, Hの全合成
  • (慶大理工)
    ○原　彰宏、森本　諒、岩崎祐樹、仮屋光馬、石川裕一、西山　繁
• Total Syntheses of Amphidinolide B, G, and H
  • Hara, A., Morimoto, R., Iwasaki, Y., Kariya, K., Ishikawa, Y., Nishiyama, S.
    (Faculty of Science and Technology, Keio University)

P-20

• (-)-エングレリンAの触媒的不斉全合成研究
  • (北大院薬)
    ○羽成泰貴、嶋田修之、穴田仁洋、橋本俊一
• Studies on Catalytic Asymmetric Synthesis of (-)-Englerin A
  • Hanari, T., Shimada, N., Anada, M., Hashimoto, S.
    (Faculty of Pharmaceutical Sciences, Hokkaido University)

P-22

• カイニン酸の全合成
  • (阪大院薬)
    ○家門拓麻、入船弥生、田中徹明、好光健彦
• Total Synthesis of Kainic Acid
  • Kamon, T., Irifune, Y., Tanaka, T., Yoshimitsu, T.
    (Graduate School of Pharmaceutical Sciences, Osaka University)

P-24

• 近赤外生物発光イメージングを目指した v-セレンテラジンの高効率合成法の開発
  • (東京医歯大^a、東工大生命理工^b、チッソ横浜研^c)
    ○隅田有人^a、飯森理絵^b、吉田　優^a、佐原由依子^c、佐藤淳一^c、井上　敏^c、細谷孝充^a,b
• Concise Synthetic Method of v-Coelenterazine Analogues Toward Near IR Bioluminescence Imaging
  • Sumida, Y.^a, Iimori, R.^b, Yoshida, S.^a, Sahara, Y.^c, Satoh, J.^c, Inouye, S.^c, Hosoya, T.^a,b
    (^aInstitute of Biomaterials and Bioengineering, Tokyo Medical and Dental University, ^bBioscience and Biotechnology, Tokyo Institute of Technology, ^cYokohama Research Center, Chisso Co.)

P-26

• C1位アルキルL-アラビノイミノフラノース誘導体の触媒的不斉合成とその生物活性評価
  • (東北薬大^a、富山大病院薬^b)
    ○名取良浩^a、今堀龍志^a、吉村祐一^a、中川進平^b、加藤　敦^b、足立伊佐雄^b、高畑廣紀^a
• Catalytic Enantioselective Synthesis and Biological Evaluation of 1-C-Alkyl-L-arabinoiminofuranose Derivatives
  • Natori, Y.^a, Imahori, T.^a, Yoshimura, Y.^a, Nakagawa, S.^b, Kato, A.^b, Adachi, I.^b, Takahata, H.^a
    (^aFaculty of Pharmaceutical Sciences, Tohoku Pharmaceutical University, ^bDepartment of Hospital Pharmacy, University of Toyama)

P-28

• ドミノ型脱離―転位―付加反応を鍵とする２－置換テトラヒドロキノリン類の合成研究：（±）―マルチネリン酸の形式合成
  • (神戸薬大)
    ○三好哲也、河井小百合、上田昌史、内藤猛章、宮田興子
• Synthetic Study on 2-Substituted Tetrahydroquinolines by Using Domino Elimination-rearrangement-addition Reaction: Formal Synthesis of (±)-Martinellic Acid
  • Miyoshi, T., Kawai, S., Ueda, M., Naito, T., Miyata, O.
    (Faculty of Pharmaceutical Science, Kobe Pharmaceutical University)

P-30

• 海綿由来血管新生阻害物質cortistatin A およびanalog化合物の合成研究
  • (阪大院薬)
    ○住井裕司、古徳直之、林　剛史、田村　理、河内崇志、森本　薫、荒井雅吉、小林資正
• Synthetic Studies and Biological Evaluation of Cortistatin A, an Anti-Angiogenic Steroidal Alkaloid from Marine Sponge, and Its Analogs
  • Sumii, Y., Kotoku, N., Hayashi, T., Tamura, S., Kawachi, T., Morimoto, K., Arai, M., Kobayashi, M.
    (Graduate School of Pharmaceutical Sciences, Osaka University)

P-32

• ビニルケトンの不斉アジリジン化とそれを鍵とするドーパミンサブタイプD₃受容体アゴニスト(+)-PD 128907の不斉形式全合成
  • (九大院理^a、I²CNER^b)
    ○内田竜也^a,b、福永恭章^a、香月　勗^b
• Catalytic Synthesis of Enantiopure Aziridinyl Ketones and Formal Asymmetric Synthesis of (+)-PD 128907
  • Uchida, T.^a,b, Fukunaga, Y.^a, Katsuki, T.^b
    (^aDepartment of Chemistry, Kyushu University, ^bInternational Institute for Carbon-Neutral Energy Research, Kyushu University)

P-34

• ルテニウム触媒によるアレンインの[2+2]環化反応を鍵工程としたWelwitindolinone A isonitrileの合成研究
  • (北大院薬)
    ○清重沙織、齋藤　望、佐藤美洋
• Synthetic Studies on Welwitindolinone A Isonitrile by Using Ruthenium-Catalyzed [2+2] Cyclization of Allenyne
  • Kiyoshige, S., Saito, N., Sato, Y.
    (Faculty of Pharmaceutical Sciences, Hokkaido University)

P-36

• 新規酵素阻害物質、ジアポルチカラシンの全合成研究
  • (慶大理工)
    ○常谷祐子、寺田大介、安蔵寿美、高尾賢一、只野金一
• Synthetic Studies of Diaporthichalasin, A New Enzyme Inhibitor
  • Tsunetani, Y., Terada, D., Anzo, T., Takao, K., Tadano, K.
    (Department of Applied Chemistry, Keio University)

P-38

• 第二世代型触媒的環化アルケニル化反応の開発と生物活性天然物合成への展開
  • (阪府大院理)
    ○竹田一貴、佐伯めぐみ、日比絢香、川合康文、豊田真弘
• Development of Second Generation Palladium-catalyzed Cycloalkenylation and Its Application to Bioactive Natural Product Synthesis
  • Takeda, K., Saeki, M., Hibi, A., Kawai, Y., Toyota, M.
    (Graduate School of Science, Osaka Prefecture University)

P-40

• 植物由来糖転移酵素を活用した高機能性配糖体の効率的合成
  • (岡山理大理^a、大分大医^b、山口大農^c、東北大工^d)
    ○濱田博喜^a、今井博也^a、北川　恵^a、下田　恵^b、小崎紳一^c、中山　亨^d
• The Synthesis of the High Functional Saponines Using Glucose Transferase Derived from Plant Cells
  • Hamada, H.^a, Imai, H.^a, Kitagawa, M.^a, Shimoda, K.^b, Ozaki, S.^c, Nakayama, T.^d
    (^aFaculty of Science, Okayama University of Science, ^bFaculty of Medicine, Oita University, ^cFaculty of Agriculture, Yamaguchi University, ^dFaculty of Technology, Tohoku University)

P-42

• 新規植物生長調整剤の開発を指向したシス桂皮酸の構造活性相関研究
  • (九大先導研^a、九大院総理工^b、農環研^c)
    ○西川慶祐^a、安部真人^a、中西一成^b、谷口智哉^b、田澤優太^b、松尾和真^b、福田　洋^b、朴　昭英^c、平舘俊太郎^c、藤井義晴^c、新藤　充^a
• The Structure-activity Relationship Study of cis-Cinnamic Acid to Develop New Plant Growth Regulator
  • Nishikawa, K.^a, Abe, M.^a, Nakanishi, K.^b, Taniguchi, T.^b, Tazawa, Y.^b, Matsuo, K.^b, Fukuda, H.^b, Park, S-Y.^c, Hiradate, S.^c, Fujii, Y.^c, Shindo, M.^a
    (^aInstitute for Material Chemistry and Engineering, Kyushu University, ^bInterdisciplinary Graduate School of Engineering Sciences, Kyushu University, ^cDepartment of Biological Safety Sciences, National Institute for Agro-Environmental Sciences)

P-44

• 海洋産アルカロイド、マンザミンBの全合成研究
  • (千葉大院薬)
    ○平岡紫陽、御原康洋、松村知亮、寺内悠樹、西田篤司
• Synthetic Study of Manzamine B
  • Hiraoka, S., Mihara, Y., Matsumura, T., Terauchi, Y., Nishida, A.
    (Graduate School of Pharmaceutical Sciences, Chiba University)

P-46

• ACAT2選択的阻害剤pyripyropene Aの構造活性相関研究ならびに全合成
  • (北里大薬^a、自治医大医^b)
    ○大多和正樹^a、松田大介^a、山崎寛之^a、大城太一^b、大村　智^a、長光　亨^a、供田　洋^a
• Total Synthesis and Structure-activity Relationship of Pyripyropene A as a ACAT2 Inhibitor
  • Ohtawa, M.^a, Matsuda, D.^a, Yamazaki, H.^a, Ohshiro, T.^b, Omura, S.^a, Nagamitsu, T.^a, Tomoda, H.^a
    (^aSchool of Pharmacy, Kitasato University/Japan, ^bDepartment of Medicine, Jichi Medical University)

P-48

• 酵母不斉還元を活用するマジンドリンAの形式全合成
  • (慶大薬^a、慶大理工^b)
    ○清水賢一^a、富田美奈^b、冨宿賢一^b、東　利則^a、須貝　威^a、庄司　満^a
• Formal Synthesis of Madindoline A Based on Yeast-mediated Asymmetric Reduction
  • Shimizu, K.^a, Tomita, M.^b, Fuhshuku, K.^b, Higashi, T.^a, Sugai, T.^a, Shoji, M.^a
    (^aFaculty of Pharmacy, Keio University, ^bFaculty of Science and Technology, Keio University)

P-50

• 抗腫瘍活性環状ペプチドサンドラマイシンの合成研究
  • (北大院薬)
    ○片山勝史、市川　聡、松田　彰
• Synthetic Study of Sandramycin
  • Katayama, K., Ichikawa, S., Matsuda, A.
    (Faculty of Pharmaceutical Sciences, Hokkaido University)

P-52

• オマエザレンの全合成
  • (北大院環境)
    ○梅澤大樹、鈴木将洋、小栗祐子、松浦裕志、沖野龍文、松田冬彦
• Total Synthesis of Omaezallene
  • Umezawa, T., Suzuki, M., Oguri, Y., Matsuura, H., Okino, T., Matsuda, F.
    (Graduate School of Environmental Science, Hokkaido University)

P-54

• (±)－Dysibetaine CPaおよび類縁体の全合成
  • (横市大院生命ナノ^a、北大院水産^b、ノースウエスタン大分子薬理生化^c)
    ○境　倫宏^a、佐々木翔太^a、石川裕一^a、酒井隆一^b、Swanson, G. T.^c、及川雅人^a
• Total Synthesis of (±)-Dysibetaine CPa and its Analogs
  • Sakai, M.^a, Sasaki, S.^a, Ishikawa,Y.^a, Sakai, R.^b, Swanson, G.^c, Oikawa, M.^a
    (^aGraduate School of Nanobioscience, Yokohama City University, ^bGraduate School of Fisheries Science, Hokkaido University, ^cMolecular Pharmacology and Biological Chemistry, Northwestern University)

P-56

• タムラミドBの合成研究
  • (岡山大院自然科学)
    ○山神雄司、岸　敬之、藤澤由佳、高村浩由、門田　功
• Synthetic Study of Tamulamide B
  • Yamagami, Y., Kishi, T., Fujisawa, Y., Takamura, H., Kadota, I.
    (Graduate School of Natural Science and Technology, Okayama University)

P-58

• α-ヒドロキシシランを用いた分子内カチオン環化反応
  • (阪市大院理)
    ○東野勝人、赤木　航、池田直子、品田哲郎、坂口和彦、大船泰史
• Cationic Intramolecular Cyclization Reaction of α-Hydroxysilane
  • Higashino, M., Akagi, W., Ikeda, N., Shinada, T., Sakaguchi, K., Ohfune, Y.
    (Graduate School of Science, Osaka City University)

P-60

• サリチルアルデヒド型イネいもち病菌毒素の合成化学的研究
  • (東北大院農^a、山形大農^b)
    ○清田洋正^a、佐々木郁香^a、田中功二^a、中村葉子^a、上田留美^a、鈴木雄二^a、桑原重文^a、貫名　学^b
• Synthetic Studies of Salicylaldehyde-type Phytotoxins Isolated from Rice Blast Fungus
  • Kiyota, H.^a, Sasaki, A.^a, Tanaka, K.^a, Nakamura, Y.^a, Ueda, R.^a, Suzuki, Y.^a, Kuwahara, S.^a, Nukina, M.^b
    (^aGraduate School of Agricultural Science, Tohoku University, ^bFaculty of Agriculture, Yamagata University)

P-62

• 抗ウイルス活性を有する新規環状デプシペプチドMA026の合成研究
  • (東理大理工^a、東理大薬^b、京府大生命環境^c)
    ○志村聡美^a、石間正浩^a、太田育恵^a、筒井悦子^a、紙透伸治^a、村田　寛^a、山崎隆之^a、鈴木孝洋^b、倉持幸司^c、竹内倫文^a、小林　進^b、菅原二三男^a
• Synthetic Studies of MA026
  • Shimura, S.^a, Ishima, M.^a, Ota, I.^a, Tsutsui, E.^a, Kamisuki, S.^a, Murata, H.^a, Yamazaki, T.^a, Suzuki, T.^b, Kuramochi, K.^c, Takeuchi, T.^a, Kobayashi, S.^b, Sugawara, F.^a
    (^aFaculty of Science and Technology, Tokyo University of Science, ^bFaculty of Pharmaceutical Science, Tokyo University of Science, ^cGraduate School of Life and Environmental Sciences, Kyoto Prefectural University)

P-64

• Lactimidomycinの全合成研究
  • (東北大院農)
    ○永沢友裕、桑原重文
• Synthetic Studies on Lactimidomycin
  • Nagasawa, T., Kuwahara, S.
    (Graduate School of Agricultural Science, Tohoku University)

P-66

• ポリ環状エーテルの収束的合成法の開発とギムノシンA合成への応用
  • (名城大薬^a、名城大院総合学術^b)
    坂井健男^a、杉本　愛^b、古川恭子^a、○森　裕二^a,b
• Convergent Synthesis of Polycyclic Ethers and Its Application to the Synthesis of Gymnocin-A
  • Sakai, T.^a, Sugimoto, A.^b, Furukawa, K.^a, Mori, Y.^a,b
    (^aFaculty of Pharmacy, Meijo University, ^bGraduate School of Environmental and Human Sciences, Meijo University)

P-68

• 立体選択的スピロケタール構築法の開発とSpirofungin A, Bの合成研究
  • (富山大院理工)
    ○宮澤眞宏、三箇剛生、榮澤　徹、村山　拓、吉原祥子、横山　初、平井美朗
• Stereoselective Synthesis of the Spiroketal Structure and Synthetic Studies of Spirofungin A and B
  • Miyazawa, M., Sanga, T., Eizawa, T., Murayama, T., Yoshihara, S., Yokoyama, H., Hirai, Y.
    (Department of Chemistry, University of Toyama)

P-70

• ブドウ由来フラボノイド配糖化酵素VvGT5、及び、VvGT6の機能解析
  • (サントリー生科財^a、サントリービジネスエキスパート^b、サントリーウエルネス^c、東北大院工^d、新潟薬大^e、立命館大生命科学^f)
    ○堀川　学^a、小埜栄一郎^b、福井祐子^c、本間　裕^d、国兼　聡^d、今井晴菜^d、高橋征司^d、中山　亨^d、石黒正路^e、河合洋介^f
• A Structure-functional Characterization of Flavonol Glycosyltransferases from Grapevines
  • Horikawa, M.^a, Ono, E.^b, Fukui, Y.^c, Homma, Y.^d, Kunikana, S.^d, Imai, H.^d, Takahashi, S.^d, Nakayama, T.^d, Ishiguro, M.^e, kawai, Y.^f
    (^aBioorganic Research Institute, Suntory Foundation for Life Sciences, ^bInstitute for Plant Science, Suntory Business Expert Limited, ^cInstitute for Health Care Science, Suntory Wellness Limited, ^dSchool of Engineering, Tohoku University, ^eApplied Life Sciences, Niigata University of Pharmacy, ^fCollege of Life Sciences, Ritsumeikan University)

P-72

• 機能未知生合成遺伝子を活用したポリケタイド系天然物の合成
  • (静岡県大薬^a、岡山大コア^b)
    ○石内勘一郎^a、中沢威人^a、大熊貴士^a、五反田康孝^a、野口博司^a、守屋央朗^b、渡辺賢二^a
• Establishing a New Methodology for Genome Mining and Biosynthesis of Natural Products through a Yeast Molecular Genomics
  • Ishiuchi, K.^a, Nakazawa, T.^a, Ookuma, T.^a, Gotanda, Y.^a, Noguchi, H.^a, Moriya, H.^b, Watanabe, K.^a
    (^aDepartment of Pharmaceutical Sciences, University of Shizuoka, ^bResearch Core for Interdisciplinary Sciences, Okayama University)